JP/EN

INOUE
RESEARCH
GROUP

ARCHIVE

Problem Session

2023年度

2023/05/06

Total Syntheses of Cephalotaxus Alkaloids (Wentao Wang)
2023/04/28

Construction of Abeo- and Diabeo-Steroid Framework from Ergosterol (Jaejoong Han)
2023/04/22

Construction of Bicyclo [3.2.1] Octane Skeleton (Yuya Shiga)
2023/04/15

Total Synthesis of Spirotryprostatins (Hiromu Kakizawa)

2022年度

2023/02/03

Works by Ullrich Jahn (Masahiro Toyoda)
2023/01/28

Construction of the Tetracyclic Core Structure of Dysiherbols (Manaka Matsumoto)
2023/01/21

Photoreactions for Constructing Fused Multicyclic Core Skeleton (Takahiro Migita)
2023/01/07

Works by John L. Wood (Shintaro Fukaya)
2022/12/24

Construction of Bicyclo[3,3,1]nonane Skeleton (Shuji Toyama)
2022/12/17

Synthetic Study of Atropurpuran and Total Synthesis of Arcutinine (Mizuki Sawada)
2022/12/10

Mutanobacin D (Aoi Takeuchi)
2022/11/19

Total Synthesis of Yuzurine-type Alkanoid Daphgraciline (Junhao Fu)
2022/11/12

Works by Ryan A. Shenvi (Yuanqi Lin)
2022/11/05

Total Synthesis Using 2+2 Cycloaddition (Yuma Komori)
2022/10/29

Synthesis of pleuromutilin analogue by S. B. Herzon (Yusuke Imamura)
2022/10/22

(Yuyan Liang)
2022/10/08

Synthetic Plan of Trichodelmol (Masanori Nagatomo)
2022/10/01

Diazo Diazirine Compound for Protein Modification (Hiroaki Itoh)
2022/09/24

Oxidative Iminium Formation (Shu Nakamura)
2022/09/17

Synthetic Plan of Grayanoids (Haruka Fujino)
2022/08/27

Site-selective acylation of glucose by organocatalysts (Yosuke Nakata)
2022/08/06

Strategy for the Construction of the Dioxaadamantane Unit of Tetrodotoxin and its Analogues (Junichi Taguchi)
2022/07/30

Total syntheses of clionastatins (Kyohei Takaoka)
2022/07/09

N-O bond (Hibiki Asai)
2022/06/24

Synthesis of Pleuromutilin (Wentao Wang)
2022/06/18

Synthetic study of rearragend limonoids (Yuuki_Watanabe)
2022/05/28

Palladium-catalyzed cascade reaction and titanocene-mediated pinacol coupling (Yuto Hikone)
2022/05/21

Total synthesis of 205B and Histrionicotoxin (Hisahiro Morozumi)
2022/05/14

Recent total synthesis by Prof. Tuoping Luo (Jaejoong Han)
2022/05/07

Works by Zhen Yang (Yuya Shiga)
2022/04/30

Total synthesis of euphorikanin A (Hiromu Kakizawa)
2022/04/23

LCMSMS analysis (Kensuke Miura)
2022/04/16

Total synthesis of preastinoids (Takahiro Watanabe)
2022/04/09

Recent total synthesis (Ayumu Watanabe)

2021年度

2022/01/29

Total synthesis of 7,20-Diisocyanoadociane and Quassin (Hisahiro Morozumi)
2022/01/22

Total synthesis of (+)-Jungermatrobrunin A (Jaejoong Han)
2022/01/13

(Yuya Shiga)
2021/12/11

Tandem cyclization (Kyohei Oga)
2021/12/03

Silicon tether approaches for regio and stereoselectivity (Junichi Taguchi)
2021/11/20

Pyridine containing Lycopodium alkaloids (Yosuke Nakata)
2021/11/13

Cephalostatin 1 (Kyohei Takaoka)
2021/11/06

3+2 cycloaddition with rhodium catalyst (Wataru Shigematsu)
2021/10/30

Galbulimima alkaloids (Hibiki Asai)
2021/10/23

Total synthesis of Avenaol and Shagene (Junhao Fu)
2021/10/09

Transformations of diterpenoid alkaloids (Koichi Hagiwara)
2021/10/02

Gold catalyzed eneyne cyclization (Haruka Fujino)
2021/09/18

Synthetic Plan of Yonarolide (Masanori Nagatomo)
2021/09/11

Total synthesis of pseudocopsinine (Takahiro Watanabe)
2021/09/04

CD spectrum (Kensuke Miura)
2021/08/28

MSbased quantitative proteomics (Aoi Takeuchi)
2021/08/21

Trans bicyclo[3.3.0]octane (Risa Yoshinaga)
2021/07/31

No title (Yuanqi Lin)
2021/07/24

NHC catalyst in total synthesis (Yuto Hikone)
2021/07/17

Lycopodium alkaloids sulfonyl rearrangement (Shu Nakamura)
2021/07/03

Total synthesis of N-methylwelwitindolinone C isothiocyanate (Yuuki Watanabe)
2021/06/12

Total Synthesis of Aspidofractinine and Lignans (Toshiya Nagai)
2021/05/29

Skeletal reorganization (Tsukasa Shimakawa)
2021/05/15

Total Synthesis of Mitrephorone A (Takumi Fukuda)
2021/05/08

Total Synthesis of marine 2,11-cyclized cembranoids (Keshu Zhang)
2021/05/01

Prediction of Protein Secondary Structure (Yun-wei Xue)
2021/04/24

Construction of 576 tricycles (Ayumu Watanabe)
2021/04/17

Calculation of dissociation constant (Koichi Kamiya)
2021/04/10

Total Synthesis of Arborisidine (Yusuke Imamura)

2020年度

2020/12/19

Concise construction of ent-kaurene and ent-beyerene type structure (Yosuke Nakata)
2020/12/12

Works by Chuang-Chuang Li (Junichi Taguchi)
2020/12/05

Total synthesis of Galanthamine Morphine (Kyohei Takaoka)
2020/11/21

Total synthesis of Melicolones AB and Caesalpinnone A (Wataru Shigematsu)
2020/11/14

Epicolactone and Preuisolactone (Hibiki Asai)
2020/11/07

CDE fragment of Aspidoserma alkaloids (Shu Nakamura)
2020/10/31

Macrocycles (Yuto Hikone)
2020/10/24

The roal of protective groups in the total synthesis of Rhodomolloanol A (Yuuki Watanabe)
2020/10/10

de novo MSMS sequencing of cyclopeptide (Aoi Takeuchi)
2020/10/03

Total Synthesis of Spongian Diterpene (Keshu Zhang)
2020/09/26

Total Synthesis of Euphorbia diterpenoid pepluanol (Junhao Fu)
2020/09/19

Total Synthesis of Waihoensene (Yuma Komori)
2020/09/12

Total Synthesis Chilocorine C (Fukuda Takumi)
2020/09/05

Total Synthesis of Caldaphnidine (Itsuki Watanabe)
2020/08/29

No title (Kensuke Miura)
2020/08/22

No title (Kotaro Tokumoto)
2020/08/01

Total Synthesis at UCB (Yinghua Wang)
2020/07/25

Synthetic Plan of Merrillianin (Masanori Nagatomo)
2020/07/18

Traditional reactions and skeletal transformation of steroids (Koichi Hagiwara)
2020/07/11

Structure Determination of Hasubanan Alkaloids (Hiroaki Itoh)
2020/07/04

Total Synthesis of herqulines (Risa Yoshinaga)
2020/06/27

Total Synthesis of Salinosporamide A (Yun-wei Xue)
2020/06/13

Total synthesis of oridonin by Luo group (Shinsuke Shimizu)
2020/06/06

Total synthesis of (–)-scabrolide A (Takahiro Watanabe)
2020/05/30

Enyne cycloisomerization (Yusuke Imamura)
2020/05/27

Total synthesis of Tetrodotoxin (Ayumu Watanabe)
2020/05/23

Dotz reaction (Daiki Kuwana)
2020/05/20

No title (Koichi Kamiya)
2020/05/16

Ring expansion/transannular reaction (Akira Hirose)
2020/05/13

Homoenolate and its equivalent in total synthesis (Tsukasa Shimakawa)
2020/05/09

Enantioselective total syntheses of cyclobutane-containing natural products (Toshiya Nagai)

2019年度

2020/02/08

Total Syntheses of Crinipellins (Yuto Hikone)
2020/01/25

Total Synthesis of Cephalotaxine (Shu Nakamura)
2020/01/11

Total Synthesis of Leuconodine Alkaloids (Aoi Takeuchi)
2019/12/21

Total Synthesis of Protoilludane Sesquiterpenes (Yuma Komori)
2019/11/30

Works by Prof. Tuoping Luo (Koichi Hagiwara)
2019/11/16

Calyciphylline-B-type Alkaloids (Koichi Kamiya)
2019/11/02

Total Synthesis of Bilobalide (Yusuke Imamura)
2019/10/26

Total Synthesis of Isomalabaricane Triterpenoids (Takahiro Watanabe)
2019/10/05

Synthetic study of spongistatin, Asymmetric synthesis of (-)-6-epi-Garcimultiflorone A (Kotaro Tokumoto)
2019/09/14

MS-based Structure Analysis (Hiroaki Itoh)
2019/09/07

Adamantane-type Natural Products (Yun-wei Xue)
2019/08/31

Synthetic Plan of Manginoid E (Masanori Nagatomo)
2019/08/03

Metathesis Cascade Reaction in Total Synthesis (Yinghua Wang)
2019/07/27

Dawei Ma's Group Synthesis (Shinsuke Shimizu)
2019/07/20

Total Synthesis by Trauner's group (Ayumu Watanabe)
2019/06/29

Application of aerobic oxidation to total synthesis (Daiki Kuwana)
2019/06/22

Construction of bicyclo [3.2.1] octane skeleton (Tsukasa Shimakawa)
2019/05/18

Cyclization (Itsuki Watanabe)
2019/05/11

Synthetic Studies Using Divinylcyclopropane (Toshiya Nagai)
2019/04/27

Chirality Transfer from Asymmetric Epoxide/Aziridine (Akira Hirose)
2019/04/13

Total Syntheses of Nyingchinoids and Merochlorin A (Takumi Fukuda)

2018年度

2019/01/12

Total synthesis of (-)-sinulariadiolide by Fürstner's group (Takahiro Watanabe)
2018/12/15

Total synthesis of FR182877 (Koichi Kamiya)
2018/12/08

Synthetic study of Isohasubanans (Yusuke Imamura)
2018/11/17

Synthetic Approaches to the trans-Fused Carotane Skeleton (Takehiro Kato)
2018/10/27

Total Syntheses by Matthew D. Shair (Takumi Fukuda)
2018/10/13

1H Chemical Shift Assignment of Peptides Using 2D NMR Experiments (Hiroaki Itoh)
2018/10/06

Reactions Including Singlet Carbene Intermediate (Tsukasa Shimakawa)
2018/09/08

Total Synthesis of Leucosceptroids, Curcumanolide A, and Anhydrochatancin (Takuya Fujiwara)
2018/09/01

Synthetic Plan of (-)-Bilobalide (Masanori Nagatomo)
2018/08/25

Reactions of Acetoxy Allenoate with Nucleophilic Catalysts (Daiki Kamakura)
2018/07/28

Total Synthesis of Astellatol, Strychnofoline and Cyclopiazonic Acid (Hiroyuki Mutoh)
2018/07/21

Asymmetric Total Synthesis of Lancifodilactone G acetate (Kosuke Minagawa)
2018/07/14

Total Synthesis of Fusarisetin A and Curcusons (Haruka Fujino)
2018/07/07

Total Synthesis of Pleuromutilin (Yuri Takada)
2018/06/30

Construction of Cembrene-based Diterpenes Core (Akira Hirose)
2018/06/16

Synthetic Studies of FR901483 (Toshiya Nagai)
2018/05/26

Total Synthesis of Sarpagine Alkaloid and kuammiline Alkaloids (Shinsuke Shimizu)
2018/04/28

Prediction of NMR Chemical Shifts (Daiki Kuwana)
2018/04/21

Synthetic Studies of Cyclocitrinol (Yinghua Wang)

2017年度

2018/03/10

Native MS Analysis (Hiroaki Itoh)
2018/03/03

Synthetic Plan of Dendrobine (Masanori Nagatomo)
2018/02/22

C-C Bond Formation Using Organoborate Reported by Prof. V. K. Aggarwal (Daiki Kamakura)
2018/01/27

Total synthesis of ent-Kauranoids (Takahiro Watanabe)
2018/01/20

Total synthesis of (-)-virosaine A (Kensuke Miura)
2018/01/11

Total Syntheses by John L. Wood (Akira Tomiyama)
2018/01/06

Miscellaneous Lycopodium Alkaloids (Yuki Fujimoto)
2017/12/22

Metal-catalyzed Cyclization of Multiynes (Akira Hirose)
2017/12/16

Synthetic Studies of Daphniphyllum Alkaloids (Kotaro Tokumoto)
2017/12/09

Total Syntheses of Spirooxindole Alkaloids (Shinsuke Shimizu)
2017/11/25

Trans-Fused 5,5 Ring (Daiki Kuwana)
2017/11/18

Total Syntheses of Xanthanolides (Yinghua Wang)
2017/10/28

Synthetic Studies of Lauroxocanes (Hiroaki Matoba)
2017/10/14

Radical Aryl Migration (Satoshi Hashimoto)
2017/09/30

Total Synthesis of Nahuoic Acid (Atsushi Hayata)
2017/09/22

Total Synthesis of Hippolachnin A (Kai Kitamura)
2017/09/16

Africanane Sesquiterpenoids (Hiroki Fujisawa)
2017/09/02

Histrionicotoxin (Yuri Takada)
2017/07/29

Synthetic approaches to the bicyclo[5.3.0]decane ring system (Takahiro Kawamata)
2017/07/22

Total Synthesis of (+)-Dictyoxetane (Kosuke Minagawa)
2017/07/15

Formal Total Synthesis of Lycojaponicumin C (Keshu Zhang)
2017/07/08

Total Synthesis of Wortmannin (Yun-wei Xue)
2017/07/01

Natural Product Including Indole Structure (Kohei Ogino)
2017/06/17

Total Syntheses of Lundurines (Takumi Fukuda)
2017/06/03

Cyclobutane and Cyclobutene Derivatives in Skeletal Rearrangement (Tukasa Shimakawa)
2017/05/27

Total Synthesis of Branimycin (Takehiro Kato)
2017/05/20

Total Synthesis of Caribenols (Yusuke Imamura)
2017/05/13

Total Synthesis of Lycodoline-Type Lycopodium Alkaloids (Benjamin Ovadia)
2017/05/06

Total Syntheses of Schisandra Nortriterpenoids (Haruka Fujino)

2016年度

2017/03/04

Total Synthesis of Echinopine A and B (Yinghua Wang)
2017/02/10

Total Synthesis of Spirotryprostatin (Yuki Fujimoto)
2017/02/03

Total Synthesis of Bolivianine and Cerorubenic Acid III (Shinsuke Shimizu)
2017/01/21

Construction of 3,4-Fused Indoles (Daiki Kuwana)
2017/01/12

Total Synthesis of Palau'amine (Yuri Takada)
2017/01/07

Synthetic study of complex meroterpenes/Total synthesis of berkeleyone A (Benjamin Ovadia)
2016/12/17

"Interrupted" reaction (Akinori Yamaguchi)
2016/12/10

Diterpene having a 5/8/5/5 ring system (Daki Kamakura)
2016/11/19

Total synthesis of (-)-Jiadifenin (Kosuke Minagawa)
2016/11/15

Total syntheses of diterpenoids posseseing bicyclo[2,2,2]octane core (Haruka Fujino)
2016/11/12

A total synthesis of (–)-6-epi-ophiobolin N (Takumi Fukuda)
2016/10/24

Tabersonine type monoterpene indole alkaloid (Tsukasa Shimakawa)
2016/10/20

Total synthesis of LicopalhineA (Koichi Kamiya)
2016/10/14

Total syntheses of asteriscanolide (Takehiro Kato)
2016/10/08

Total syntheses of Maoecrystal V (Yusuke Imamura)
2016/09/24

Tetrahydrothiophene (Hiroaki Itoh)
2016/09/10

Construction of bridged cyclobutane (Masanori Nagatomo)
2016/09/03

Total Syntheses of Pallmbins (Hiroaki Matoba)
2016/08/27

Total synthesis of coriolin (Yuki Nakagawa)
2016/08/06

Total synthesis of jiadifenolide (Koichi Hagiwara)
2016/07/23

STR-8 and GA3 (Satoshi Hashimoto)
2016/07/16

Total synthesis of periconiasin and rubialatin (Atsushi Hayata)
2016/07/09

Biomimetic Total Synthesis of Dimeric Phenylethanoids (Atsushi Hayata)
2016/07/04

Strategies for the synthesis of leucosceptroids (Takahiro Kawamata)
2016/06/25

Recent total synthesis of monoterpene indole alkaloids (Eiji Yoshida)
2016/06/18

Reaction of vinyl sulfide in total synthesis (Keisuke Masuda)
2016/06/04

Azocine and Azocane (Shun Yoshioka)
2016/05/30

Synthetic Studies of Englerin A (Hiroki Fujisawa)
2016/05/21

Total synthesis of Pactamycin (Hideyuki Sawada)
2016/05/14

Total synthesis of (-)-lingzhiol (Komei Sakata)
2016/05/07

Synthetic Study of indoxamycins (Masaki Koshimizu)
2016/04/30

Glucosepane (Takuya Kaji)
2016/04/09

Titanacyclopropane (Shunichiroh Katoh)

2015年度

2016/03/05

Transformation of Isoxazoles (Hiroaki Itoh)
2016/02/27

Studies toward Total Synthesis of Ryanodine (Masanori Nagatomo)
2016/02/05

Recent Remarkable Chemistry Related to Pyrrole (Kai Kitamura)
2016/01/23

Total syntheses by Prof. R. Hong group (Hiroaki Matoba)
2016/01/14

Total synthesis of Alsmaphorazine B, (-)-Dendrobine and Huperizine A (Hiroki Fujisawa)
2016/01/09

Total Synthesis of Pallavicinin and Neopallavicinin (Koichi Hagiwara)
2015/12/12

Synthesis of Seven-Membered-Ring Carbamates etc. (Satoshi Hashimoto)
2015/11/28

Stereoselective Construction of Skipped Polyol and Polymethyl Structural Motif (Masaki Koshimizu)
2015/11/20

Total synthesis of Samaderine (Daiki Kamakura)
2015/11/14

Collective Total Synthesis of Atisane-Type Diterpenes and Atisine-Type Diterpenoid Alkaloids (Komei Sakata)
2015/11/07

A total synthesis of (+)-artemisinin by S. P. Cook et al. (Yuki Fujimoto)
2015/10/16

A total synthesis of (-)-Acutumine by Herzon’s group (Kotaro Tokumoto)
2015/10/09

Chemistry around Onium Ylide (Yuki Matsui)
2015/10/02

A Total Synthesis of ( )-Basiliolide B by Lee et al. (Daiki Kuwana)
2015/09/26

Total Synthesis of Limonin (Yinghua Wang)
2015/09/12

(Hirotatsu Umihara)
2015/09/12

Transfer of various chiralites (Kengo Masuda)
2015/08/01

α,α-Disubstituted amino acids (Atsushi Hayata)
2015/07/25

Dead End and Detours (Haruka Fujino)
2015/07/04

Synthesis of 2,8-dioxabicyclo[3,2,1]octane skeleton (Keisuke Masuda)
2015/06/27

Wittig Rearrangement (Shun Yoshioka)
2015/06/13

Transannular reaction and rearrangement related to trans-cycloalkenes (Takahiro Kawamata)
2015/05/29

First total synthesis of steenkrotin A (Kosuke Minagawa)
2015/05/23

Total synthesis of (+)-Scholarisine A (Hideyuki Sawada)
2015/05/16

Total synthesis of phomactin A by Hsung (Akinori Yamaguchi)
2015/05/09

Orbital symmetry and Woodward-Hoffmann rules (Shunichiroh Katoh)
2015/04/24

Enterocin (Takuya Kaji)
2015/04/18

Azetidine (Tomoya Yamashita)
2015/04/11

Molecular orbital theory and Hartree-Fock method- (Yuki Nakagawa)

Literature Seminar

2023年度

2023/05/20

Photocatalytic [2+2]-Cycloaddition Using StyrenylBpin (Yuto Hikone)
2023/05/06

Microwave Effect (Shu Nakamura)
2023/04/22

Real Time Analysis of Protease Reaction (Aoi Takeuchi)
2023/04/15

Csp3-Csp3 Cross-Coupling Using Alcohol and Alkyl Bromide (Yuma Komori)
2023/04/08

Isoxazole Photo-Cross-Linker (Junhao Fu)

2022年度

2023/01/21

B(C6F5)3-Mediated Iminium Ion Formation (Koichi Hagiwara)
2022/12/24

Targeting Recruitment Self Assembly Strategy (Yuanqi Lin)
2022/12/10

Synthesis of Nonclassical Taxane (Wentao Wang)
2022/11/19

Total Syntheses of Mannopeptimycins (Takahiro Migita)
2022/11/12

Total Synthesis of Grayanane Diterpenoids (Masahiro Toyoda)
2022/11/05

Total Syntheses of Ginkgolide A B C (Shintaro Fukaya)
2022/10/29

Total Synthesis of Conidiogenones and Aberrarone (Manaka Matsumoto)
2022/10/08

Total Synthesis of Myrioneurinol (Mizuki Sawada)
2022/10/01

Total syntheses of Calyciphylline A-Type Alkaloids (Shuji Toyama)
2022/09/24

Development of an effective extension method of carbon chain using new boronates (Hisahiro Morozumi)
2022/09/10

Metallaphotoredox Fragment Couplings of Alcohols and Carboxylic Acids (Jaejoong Han)
2022/08/27

Surrogate Asymmetric Mannich Reaction with Sulfinimines and Stereodivergent Olefination with Sulfur Ylides (Yuya Shiga)
2022/08/06

Prediction of the Passive Membrane Permeability of Molecules (Hiromu Kakizawa)
2022/07/23

SmI2-catalyzed reaction by Procter's group (Takahiro Watanabe)
2022/07/16

Ferroptosis Inducer (Kensuke Miura)
2022/07/09

Functionalization of BC-ring of daphnane and tigliane diterpenes (Ayumu Watanabe)
2022/06/18

Asymmetric Total Synthesis of Norzoanthamine (Yuyan Liang)
2022/05/28

Development of Next Generation Taxoids by Iwao Ojima (Yosuke Nakata)
2022/05/07

Access to β- and γ-Lactams via Olefin Difunctionalization (Junichi_Taguchi)
2022/04/30

Steric Repulsion and London Dispersion (Kyohei_Takaoka)
2022/04/23

Carbonyl 1,2-transposition (Kyohei Oga)
2022/04/16

Chemical recycling of polystyrene (Wataru Shigematsu)
2022/04/09

Enolization using NaHMDS (Hibiki Asai)

2021年度

2022/01/08

In-Depth Understanding of Chemical Reactivity (Haruka Fujino)
2021/12/25

1H NMR (GEMSTONE) (Yuuki Watanabe)
2021/12/11

Conformational Analysis for Lectin-Glycan Recognition (Aoi Takeuchi)
2021/12/03

Photoaffinity Labeling Preferences of Diazirines (Lin Yuanqi)
2021/11/20

Total Synthesis of Vancomycin Aglycon by Boger Group (Yuto Hikone)
2021/11/13

Tertiary dialkyl ether synthesis (Risa Yoshinaga)
2021/11/06

Chemical characters of Db (Shu Nakamura)
2021/10/30

Single Electron Reduction of Aryl Halides Using Radical Anion (Yuma Komori)
2021/10/09

Total Synthesis of Altemicidin and SB-203207 (Jaejoong Han)
2021/10/02

Synthesis And Bioactivity of Albicidin Analogues (Hiromu Kakizawa)
2021/09/25

Total Synthesis of Spiroxin A C D (Yuya Shiga)
2021/09/18

Total syntheses of Hetisine-Type Diterpenoid Alkaloids (Hisahiro Morozumi)
2021/09/04

Radical reactions using α-aminoalkyl radicals (Toshiya Nagai)
2021/08/28

From electrocatalysis to electrophotocatalysis (Tsukasa Shimakawa)
2021/08/21

Pyridone Ligand-Accelerated C-H Functionalization (Takumi Fukuda)
2021/07/24

DNA as Storage Medium (Yunwei Xue)
2021/07/17

Selective functionalization of Carbohydrates (Ayumu Watanabe)
2021/07/03

β-C-H Alkylation of Carbonyls (Yusuke Imamura)
2021/06/19

Total Synthesis of (±)-Cephanolides (Kyohei Oga)
2021/06/12

Synthesis and Application of B-N Containing Tryptophan (Yosuke Nakata)
2021/05/29

Skeletal Editing through Direct Nitrogen Deletion of Secondary Amines (Junichi Taguchi)
2021/05/22

Asymmetricchlorination (Kyohei Takaoka)
2021/05/15

Coupling of Allyl Triflate with Allyl Tosylate (Wataru Shigematsu)
2021/05/08

Direct Asymmetric Vinylogous Mannich Reaction (Hibiki Asai)
2021/05/01

Tunable methacrylamides as new eletrophile for cystein targeted covalent inhibitors (Junhao Fu)
2021/04/24

Hydration of nitriles with Ghaffar-Parkins catalyst (Takahiro Watanabe)
2021/04/17

Inhibitors of Drug Resistant EGFR Mutant (Kensuke Miura)

2020年度

2020/11/21

Molecular Complexity (Masanori Nagatomo)
2020/11/14

Deaminative Radical Formation of Primary Amine (Koichi Hagiwara)
2020/10/31

Total Synthesis of Taxol (Yusuke Imamura)
2020/10/24

The liver brain gut neural arc (Ayumu Watanabe)
2020/10/10

Catalyst Design Using Machine Learning (Junichi Taguchi)
2020/10/03

Substrate Directed Peptide Synthesis with Lewis Acid (Yosuke Nakata)
2020/09/26

Hydroamination (Kyohei Takaoka)
2020/09/19

Total Synthesis of (-)-Epicoccin G and (-)-Rostratin A (Wataru Shigematsu)
2020/09/12

Total Synthesis of (+)-Corymine (Hibiki Asai)
2020/09/05

Total Synthesis of Pallambins (Risa Yoshinaga)
2020/08/29

Cu(III) OtBu with phosphine (Shu Nakamura)
2020/08/01

Photoexited-State Pd Catalysis (Takumi Fukuda)
2020/07/18

DNA Encoded Library (Aoi Takeuchi)
2020/06/27

Hypervalent Iodine Catalyzed Enantioselective Acetoxylation of Ketone (Yuma Komori)
2020/06/13

Carbonyl alkylative amination (Keshu Zhang)
2020/05/30

affinity probe and chemical proteomics (Koichi Kamiya)
2020/05/20

Asymmetric Cu-Catalyzed C(sp3)-C(sp) Coupling by Liu’s group (Toshiya Nagai)
2020/04/25

Rational design of Pd and Ni catalyst for the efficient C-N bond formation reaction (Tsukasa Shimakawa)
2020/04/11

Cerium Catalyzed Functionalization by Zhiwei Zuo group (Shinsuke Shimizu)

2019年度

2020/01/25

Dinickel Catalyst with Redox Active Ligand (Koichi Hagiwara)
2020/01/11

Mn Catalyzed Redox Cascade Reaction (Yuuki Watanabe)
2019/12/07

Total Synthesis of (-)-Vinigrol (Yuto Hikone)
2019/11/30

Total Synthesis of (-)-Jorumycin (Shu Nakamura)
2019/11/16

Designing an Organocatalyst-Driven Peptide Synthesis (Aoi Takeuchi)
2019/11/02

Total Synthesis of TAN-1085 (Komori Yuma)
2019/10/05

Multivalent Interactions (Kensuke Miura)
2019/07/07

Application of DNA self-assembly (Akira Hirose)
2019/06/29

Photochirogenesis using photosensitizers (Takahiro Watanabe)
2019/06/22

α-Fluorination of amide and stereodivergent synthesis of 1,4-dicarbonyls by Nuno Maulide’s group (Toshiya Nagai)
2019/05/18

Carbon Dioxide Mediated Arylation of Amine (Shinsuke Shimizu)
2019/04/13

Carbonyl Olefin Metathesis (Yinghua Wang)

2018年度

2019/01/12

Works by Prof. Bill Morandi -Isofunctional Reactions- (Koichi Hagiwara)
2019/01/05

Siderophores and Metallophores (Hiroaki Itoh)
2018/12/22

De novo Designed Antimicrobial Capsids (Takuya Fujiwara)
2018/12/15

Metal Catalyzed Asymmetric Cross Coupling Reactions (Daiki Kamakura)
2018/11/10

Photocatalytic Bioconjugation of Native Proteins (Kosuke Minagawa)
2018/10/27

Strained Olefin Catalysts (Haruka Fujino)
2018/08/25

Scaffold Protein Gephyrine (Kensuke Miura)
2018/07/21

Photochromic Fluorescent Probe (Takehiro Kato)
2018/07/14

Design of Enzyme (Yun-wei Xue)
2018/06/30

Asymmetric Brønstedacid catalysisdeveloped by Benjamin List's group (Tsukawa Shimakawa)
2018/06/16

Library Strategy for Cyclic Peptide (Koichi Kamiya)
2018/05/26

Ketone α C-H Alkylation with Alkenes (Takumi Fukuda)
2018/04/28

Catalytic Enantioselective Fluorination of Alkene (Takahiro Watanabe)
2018/04/21

Predicting Reaction Performance Using Machine Learning(Yusuke Imamura)

2017年度

2018/03/03

Probing into RNA Structures (Yun-wei Xue)
2018/02/10

Remote C-H Functionaliation of Amines (Takumi Fukuda)
2018/01/27

Efficient Electrocatalytic Reduction of CO2 (Takehiro Kato)
2018/01/11

Photoinduced C-N Cross Coupling Reaction Developed by G. C. Fu’s Group (Tsukasa Shimakawa)
2018/01/06

New Madelalides Expand Macrolide Series of Mitochondrial Inhibitors (Koichi Kamiya)
2017/12/22

Total Syntheses of illicium Sesquiterpenes (Kohei Ogino)
2017/12/16

Glycocalyx Engineering (Hiroaki Itoh)
2017/12/09

Dearomatization of Benzene Ring (Yusuke Imamura)
2017/11/25

DNA-encoded Library (Yuri Takada)
2017/11/18

Coupling Reactions Using Excited State Organonickel Complex (Daiki Kamakura)
2017/10/28

Prof. Ang Li (Kosuke Minagawa)
2017/10/07

Construction of Polyketides Bearing Bridgehead Diols(Haruka Fujino)
2017/09/30

Synthetic Methodology for Tetrodotoxin (Takahiro Watanabe)
2017/09/22

Phosphorothioate_oligonucleotides (Kensuke Miura)
2017/09/16

Total Syntheses of Huperzine Q (Akira Tomiyama)
2017/09/02

Total Synthesis of Calicheamicin Type Enediyne Natural Products (Yuki Fujimoto)
2017/08/26

CO-Surrogate (Benjamin Ovadia)
2017/07/29

Artificial Tail-to-Head Terpene Cyclization (Akira Hirose)
2017/07/22

Ligand-Based De Novo Drug Design (Kotaro Tokumoto)
2017/07/15

Stereoselective Transfer Hydrogenation of Alkynes to Alkene (Shinsuke Shimizu)
2017/07/08

Radical Conjugate Addition (Daiki Kuwana)
2017/07/01

Nugent Reagent -Application for Radical Reactions- (Yinghua Wang)
2017/06/17

Total Synthesis of Pleuromutilin (Hiroaki Matoba)
2017/06/03

Synthesis of Diols by Site Selective Oxidation of Alcohols (Hiroki Fujisawa)
2017/05/27

Salinomycin Kills Cancer Stem Cells by Sequestering Iron in Lysosomes (Atsushi Hayata)
2017/05/20

Electrochemical Alcohol Oxidation Mediated by Nitroxyl Radicals (Satoshi Hashimoto)
2017/05/13

MicroRNA Therapeutics -Overview and Cutting Edge of Small Molecule-based Approach- (Kai Kitamura)

2016年度

2017/03/22

Rethinking Library Strategy for Drug Discovery (Hiroaki Itoh)
2017/02/08

Spongistatin-based Anti-cancer Agent (Daisuke Urabe)
2017/02/03

Cross-Electrophile Coupling (Daiki Kamakura)
2017/01/27

Total Synthesis of Morphine (Takumi Fukuda)
2017/01/21

Integration of C-C Bond Activation and C-H Bond Activation (Tsukasa Shimakawa)
2016/12/17

Construction of contiguous quaternary carbon (Yusuke Imamura)
2016/12/10

Peptide stapling via C-H activation (Hiroaki Matoba)
2016/11/26

Coupling Reaction Using N-tosylhydrazone as The Precursor of Diazo Compound (Hiroki Fujisawa)
2016/11/19

Chemistry around 1,1-Diborylalkanes (Koichi Hagiwara)
2016/11/15

Antibody Drug Conjugates (Satoshi Hashimoto)
2016/11/12

CPPs and Its Application to DM1 (Atsushi Hayata)
2016/10/24

Dehydro Diels Alder Reaction (Takahiro Kawamata)
2016/10/20

Chemical Manipuration of Protein Functions (Kai Kitamura)
2016/10/14

Total synthesis of Isoschizogamine (Eiji Yoshida)
2016/10/08

Chemistry of Hellicene (Keisuke Masuda)
2016/09/24

Proton Coupled Electron Transfer (Shun Yoshioka)
2016/09/16

Computer-Assisted Synthetic Planning the End of the Beggining (Yuki Nakagawa)
2016/09/10

Chemistry around Cubane and its Derivatives (Hideyuki Sawada)
2016/09/03

Biomimetic Synthesis of Dibefurin and Epicolactone (Komei Sakata)
2016/08/29

Endogenous Lipid Mediators (Daisuke Urabe)
2016/08/27

Selectfluor mediated Organic Synthesis (Masaki Koshiomizu)
2016/08/06

Designing Folded Structure (Takuya Kaji)
2016/07/23

Active Learning in Drug Discovery (Shunichiroh Katoh)
2016/07/16

Reactions of Pyrone (Yinghua Wang)
2016/07/09

Total Synthesis of Solithromycin (Shinsuke Shimizu)
2016/07/04

Total Synthesis of Callipeltosides A-C (Yuki Fujimoto)
2016/06/25

Total Synthesis of Saxitoxin (Akira Hirose)
2016/06/18

Application of Mechanoresponsive Polymer to Drug Delivery (Daiki Kuwana)
2016/06/04

Protein Bioconjugation Using π-clamp (Kotaro Tokumoto)
2016/05/30

Search a new antibiotic kills pathogens without detectable resistance (Yuri Takada)
2016/05/21

Photoredox Catalysis (Benjamin Ovadia)
2016/05/14

Hydroamination (Akinori Yamaguchi)
2016/05/07

Anion-π Catalysis (Hiroyuki Mutoh)
2016/04/30

Stereoinversion of tertiary alcohols to tertiary-alkyl isonitriles and amines (Kosuke Minagawa)
2016/04/09

Solid supported organometallic catalysts (Haruka Fujino)

2015年度

2016/03/05

Total synthesis of merrilactone (Hirotatsu Umihara)
2016/02/27

Total synthesis of gelsemine (Yuki Fujimoto)
2016/02/05

Loss of function (Kotaro Tokumoto)
2016/01/30

Total Synthesis of Enigmazole (Daiki Kuwana)
2016/01/23

Total Syntheses of Schindilactone A and Rubriflordilactone A (Yinghua Wang)
2016/01/14

Voltage-sensitive_Probes (Atsushi Hayata)
2016/01/09

Diterpenoid alkaloids (Daiki Kamakura)

研究年報